VolSurf+ user manual


Table of Contents
1. Overview
1.1. What is VolSurf+?
1.2. Program citation
1.3. Program organization
1.4. Limitations
2. What is new in VolSurf+?
2.1. New Modules in VolSurf+
2.2. New descriptors
2.3. Standard library models
2.4. Automatic Protonation-Deprotonation
2.5. Handling of SMILES structure or 2D SD files
2.6. Handling of a large series of compounds
2.7. User settings
2.8. Independence from the operating system
2.9. New and more flexible command line interface
3. Installation
3.1. Installation of the Windows version
3.2. Installation of the UNIX version
3.2.1. Installing VolSurf+ on a NFS server
4. Background
4.1. 3D maps
4.2. From 3D maps to 2D descriptors
4.3. Multivariate analysis of VolSurf+ descriptors
4.4. References
5. VolSurf+ Descriptors
5.1. Overview
5.2. Details
5.2.1. Size and shape descriptors
5.2.2. Descriptors of hydrophilic regions
5.2.3. Descriptors of hydrophobic regions
5.2.4. INTEraction enerGY (= INTEGY) moments
5.2.5. Descriptors of H-bond donor / acceptor regions
5.2.6. Mixed descriptors
5.2.7. Charge State descriptors
5.2.8. 3D pharmacophoric descriptors
5.2.9. ADME model descriptors
5.3. Conclusions
6. VolSurf+ ADME descriptors
6.1. Blood-Brain Barrier permeation model (LogBB)
6.2. Thermodynamic solubility model (SOLY)
6.3. Caco2 permeation model (CACO2)
6.4. Protein Binding model (PB)
6.5. Volume of Distribution model (VD)
6.6. CYP3A4 Metabolic Stability model (MetStab)
7. Statistical Tools
7.1. Principal Components Analysis (PCA)
7.1.1. Uses of PCA
7.2. Consensus PCA
7.2.1. Uses of CPCA
7.3. Partial Least Squares (PLS)
7.3.1. PLS modeling
7.3.2. Tests of predictive ability: Cross-validation
7.3.3. Uses of PLS
7.4. References
8. Modeling data
8.1. PCA model generation
8.2. External PCA projection
8.3. CPCA model generation
8.4. PLS model generation
8.5. Validation of the PLS model
8.6. External PLS prediction
8.7. Projection on library model
8.8. Select subset
9. Command-line interface
9.1. Introduction
9.2. Keywords
9.2.1. General keywords
9.2.2. Constants (VSL_constant)
9.2.3. Parameters (VSL_param)
9.3. Strings (VSL_string)
9.4. VSL statements
9.4.1. File statements
9.4.2. Import statements
9.4.3. Datamatrix Export statements
9.4.4. Configure statements
9.4.5. Modeling statements
9.4.6. Selector statements
10. Overview of the program GRID
10.1. Energy functions of program GRID
10.1.1. The Lennard-Jones potential
10.1.2. The electrostatic potential
10.1.3. The hydrogen bond potential
10.1.4. The entropy term
10.2. VolSurf+ Probes

Latest versions

Login

Username

Password

Register | Lost password?