MetaSite user manual

Gabriele Cruciani

Riccardo Vianello

Ismael Zamora

Edited by

Gianluca Sforna

Paolo Benedetti


Table of Contents
1. Overview
1.1. What is MetaSite?
1.2. MetaSite features
1.3. What MetaSite is not?
1.4. Program citation.
1.5. Program organization
1.6. Limitations.
1.7. User's support.
2. Background
2.1. Introduction
2.2. Protein Treatment
2.3. 3D structure of substrates, and fingerprint generation
2.4. Substrate-CYP enzyme comparison: the Recognition component
2.5. The Reactivity component
2.6. Computation of the probability of site of metabolism
2.7. Conclusions
2.8. References
3. Installation
3.1. Installation of the windows version
3.2. Installation of the unix version
3.2.1. Installing MetaSite on a NFS server
3.2.2. Editing the launch scripts
4. Command line options
4.1. Examples
5. MetaSite menu bars
5.1. File menu
5.1.1. Open/Open ascii
5.1.2. Close
5.1.3. Save
5.1.4. Save As/Save_As_Ascii
5.1.5. Export As SD File
5.1.6. Exit
5.2. MetaSite menu
5.2.1. Sketch substrate
5.2.2. Load substrates as single conformers
5.2.3. Load substrates as conformer sets
5.2.4. Enter SMILES string
5.2.5. Load SMILES list
5.2.6. Run site of metabolism prediction
5.2.7. Evaluate inhibition
5.2.8. Tabulate
5.3. View menu
5.3.1. 2D View
5.3.2. Substrate rendering
5.3.3. Atoms color
5.3.4. Sort histograms
5.3.5. Reactivity correction
5.3.6. Tool bar
5.3.7. Status bar
5.3.8. Interface Style
5.4. CYP menu
5.4.1. Import enzyme
5.5. Help menu
6. MetaSite tutorial
6.1. Case study 1. Direct editing of substrate structures.
6.2. Case study 2. Input of Salmeterol as single conformation file.
6.3. Case study 3. Comparing common reactivity criteria and metabolic reactivity.
6.4. Case study 4. Prediction results using different cytochrome models on the same substrates structures.
6.5. Case study 5. MetaSite applications.
6.6. Case study 6. Running MetaSite from the command line
6.7. Conclusions
A. Sketching small molecules
A.1. Get starting
A.2. Atom types
A.3. 3D converting procedure
A.4. Toolbar items and controls
A.4.1. Clear document
A.4.2. Undo/Redo
A.4.3. Change atom type
A.4.4. Insert bond
A.4.5. Increase/Decrease charge
A.4.6. Select
A.4.7. Move
A.4.8. Rotate
A.4.9. Delete
A.4.10. Group/Ungroup
A.4.11. Select all
A.4.12. Show atom colors
A.4.13. Show warnings
A.4.14. Show explicit hydrogens
A.4.15. Implicit hydrogens
A.4.16. Zoom

Latest versions

Login

Username

Password

Register | Lost password?